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Ku ya 15 Mata 2022, icyitegererezo cy’icyuma cya hydrocloride ya Lecardipine cyarangiye icyarimwe, kandi ubu umusaruro ni 5Mt / ukwezi.

Ku ya 15 Mata 2022, icyitegererezo cy’icyuma cya hydrocloride ya Lecardipine cyarangiye icyarimwe, kandi ubu umusaruro ni 5Mt / ukwezi.
Izina ry'icyongereza:Lercanidipine hydrochloride
Izina ryimiti:1,4-Dihydro-2,6-dimethyl-4- (3-nitrophenyl) -3,5-pyridinedicarboxylic aside 2 - [(3,3-di phenylpropyl) methylamino] -l, l-dimethylethyl methyl ester hydrochloride.

URUBANZA No: 132866-11-6
Gusaba:Mu kuvura imiti ya hydrochloride ya Lecardipine, ntabwo bizagira ingaruka mbi ku maraso ya glucose na lipide, kandi bigira ingaruka zikomeye zo kurwanya umuvuduko ukabije.

Icyizere cy'isoko :
Mu Bushinwa hari abarwayi barenga miliyoni 200 barenga umuvuduko ukabije, kandi buri mwaka hari abarwayi bashya bafite umuvuduko ukabije wa miliyoni 10, abenshi muri bo bakaba batagenzurwa, bigatuma habaho ibibazo byinshi by’indwara ziterwa na hypertension nka stroke, ndetse n’urupfu buri mwaka mu Bushinwa Muri 3 miliyoni z'abarwayi bafite indwara z'umutima-damura, 50% zifitanye isano na hypertension, kandi buri mwaka amafaranga yo kuvura indwara z'umutima-damura agera kuri miliyari 309.8.Impamvu yo kugenzura nabi ntabwo ari uko abarwayi bakeneye kumenya hypertension ningaruka zayo bigomba kunozwa gusa, ahubwo ni uko abarwayi benshi bakeneye gufata imiti ubuzima bwabo bwose batubahiriza amategeko kandi ntibashobora gufata imiti buri munsi Ariko, ibi birerekana kandi ko isoko ryibiyobyabwenge birwanya umuvuduko ukabije.Ugereranije nibiyobyabwenge bisa, hydrochloride ya lokarbodipine ifite imitsi ihitamo.Imiterere yihariye ya lipofilique ituma itinda kandi iramba ya antivypertensique Ingaruka ya aterogeneque, cyane cyane ibereye abarwayi ba hypertension barwaye aterosklerose, ifite agaciro gakomeye k’amavuriro kandi ifite isoko ryagutse.

Igikorwa cya farumasi :
Lecardipine ni igisekuru gishya cya dihydropyridine calcium umuyoboro witsinda hystereze, hamwe noguhitamo gukomeye kwamaraso, ingaruka zoroheje, ingaruka zikomeye zo kurwanya umuvuduko ukabije, igihe kirekire cyibikorwa, ingaruka mbi za inotropique nibindi.Mu bushakashatsi bwa vitro bwerekanye ko locarbodipine igira ingaruka zitaziguye ku mitsi yoroshye yimitsi itwara imitsi, bityo ikaba ifite ingaruka zikomeye zo kurwanya umuvuduko ukabije muri vivo, ariko ntigire ingaruka nke ku mutima no ku mutima.Kubera gene nini ya hydrophobique hamwe no gukomera kwa lipide, locarbodipine ikwirakwizwa vuba mumyanya ningingo nyuma yo kwinjira mumubiri, igahuza cyane ningirangingo yimitsi itwara imitsi, hanyuma ikarekura buhoro.Kubwibyo, nubwo serumu yibi biyobyabwenge ifite igihe gito cyo kurandura igice cyo kunanirwa, ingaruka zayo ziramba.


Igihe cyo kohereza: Apr-15-2022